Synthesis and Antiprotozoal Activity of N-Alkoxy Analogues of the Trypanocidal Lead Compound 4,4′-Bis(imidazolinylamino)diphenylamine with Improved Human Blood−Brain Barrier Permeability-Reference-Cited by-同舟云学术

Synthesis and Antiprotozoal Activity of N-Alkoxy Analogues of the Trypanocidal Lead Compound 4,4′-Bis(imidazolinylamino)diphenylamine with Improved Human Blood−Brain Barrier Permeability

Published:2010-12-22 Issue:2 Volume:54 Page:485-494
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nieto Lidia¹,Mascaraque Ainhoa¹,Miller Florence²³,Glacial Fabienne²³,Ríos Martínez Carlos¹,Kaiser Marcel⁴⁵,Brun Reto⁴⁵,Dardonville Christophe¹

Affiliation:

1. Instituto de Química Médica, CSIC, Juan de la Cierva 3, E-28006 Madrid, Spain

2. Institut Cochin, Université Paris Descartes, CNRS (UMR 8104), Paris, France

3. Inserm, U1016, Paris, France

4. Swiss Tropical and Public Health Institute, Socinstrasse 57, CH-4002 Basel, Switzerland

5. University of Basel, Basel, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm101335q

Reference53 articles.

1. Human African Trypanosomiasis: Global View.http://www.dndi.org/diseases/hat/global-view.html(accessed 25th November 2009) .

2. WHO. Control and Surveillance of African Trypanosomiaisis;WHO Technical Report Series, Vol.881;World Health Organization:Geneva, 1998; pp1−113.

3. Human African trypanosomiasis, chemotherapy and CNS disease

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