Synthesis, Radiosynthesis, and Biological Evaluation of Carbon-11 and Fluorine-18 (N-Fluoroalkyl) Labeled 2β-Carbomethoxy-3β-(4'-(3-furyl)phenyl)tropanes and -nortropanes: Candidate Radioligands for in Vivo Imaging of the Serotonin Transporter with Positron Emission Tomography-Reference-Cited by-同舟云学术

Synthesis, Radiosynthesis, and Biological Evaluation of Carbon-11 and Fluorine-18 (N-Fluoroalkyl) Labeled 2β-Carbomethoxy-3β-(4'-(3-furyl)phenyl)tropanes and -nortropanes: Candidate Radioligands for in Vivo Imaging of the Serotonin Transporter with Positron Emission Tomography

Published:2005-10-04 Issue:22 Volume:48 Page:7080-7083
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Stehouwer Jeffrey S.¹,Plisson Christophe¹,Jarkas Nachwa¹,Zeng Fanxing¹,Voll Ronald J.¹,Williams Larry¹,Martarello Laurent¹,Votaw John R.¹,Tamagnan Gilles¹,Goodman Mark M.¹

Affiliation:

1. Department of Radiology, Emory University, 1364 Clifton Road NE, Atlanta, Georgia 30322, and Department of Psychiatry, Yale University, West Haven Connecticut 06516

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0504095

Reference18 articles.

1. A novel class of calcium-entry blockers: the 1-[[4-(aminoalkoxy)phenyl]sulfonyl]indolizines

2. Chemistry, Design, and Structure−Activity Relationship of Cocaine Antagonists

3. 2002 Medicinal Chemistry Division Award Address: Monoamine Transporters and Opioid Receptors. Targets for Addiction Therapy

4. N-Substituted Analogs of 2β-Carbomethoxy-3β-(4‘-iodophenyl)tropane (β-CIT) with Selective Affinity to Dopamine or Serotonin Transporters in Rat Forebrain

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