Novel Conformationally Constrained Tropane Analogues by 6-endo-trig Radical Cyclization and Stille Coupling − Switch of Activity toward the Serotonin and/or Norepinephrine Transporter-Reference-Cited by-同舟云学术

Novel Conformationally Constrained Tropane Analogues by 6-endo-trig Radical Cyclization and Stille Coupling − Switch of Activity toward the Serotonin and/or Norepinephrine Transporter

Published:2000-05-01 Issue:10 Volume:43 Page:2064-2071
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hoepping Alexander¹,Johnson Kenneth M.¹,George Clifford¹,Flippen-Anderson Judith¹,Kozikowski Alan P.¹

Affiliation:

1. Drug Discovery Program, Georgetown University Medical Center, 3900 Reservoir Road, NW, Washington, D.C. 20007-2197, Department of Pharmacology and Toxicology, University of Texas Medical Branch, Galveston, Texas 77555-1031, and Laboratory for the Structure of Matter, Code 6030, Naval Research Laboratory, 4555 Overlook Avenue, SW, Washington, D.C. 20375-5000

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0001121

Reference33 articles.

1. Serotonergic mechanisms involved in the discriminative stimulus, reinforcing and subjective effects of cocaine

2. Changes in serotonin and norepinephrine uptake sites after chronic cocaine: pre- vs. post-withdrawal effects

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