The Taming of Capsaicin. Reversal of the Vanilloid Activity of N-Acylvanillamines by Aromatic Iodination-Reference-Cited by-同舟云学术

The Taming of Capsaicin. Reversal of the Vanilloid Activity of N-Acylvanillamines by Aromatic Iodination

Published:2005-06-10 Issue:14 Volume:48 Page:4663-4669
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Appendino Giovanni¹,Daddario Nives¹,Minassi Alberto¹,Moriello Aniello Schiano¹,De Petrocellis Luciano¹,Di Marzo Vincenzo¹

Affiliation:

1. Dipartimento di Scienze Chimiche, Alimentari, Farmaceutiche e Farmacologiche, Via Bovio 9, 28100 Novara, Italy; Endocannabinoid Research Group, Institute of Biomolecular Chemistry, CNR, Via Campi Flegrei 34, 80078 Pozzuoli (NA), Italy, Endocannabinoid Research Group, Istitute of Cibernetica “Eduardo Caianiello”, CNR, Via Campi Flegrei 34, 80078 Pozzuoli (NA)

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050139q

Reference37 articles.

1. Vanilloid Receptor Ligands

2. Biochemical pharmacology of the vanilloid receptor TRPV1. An update

3. TRPV1 (vanilloid receptor, capsaicin receptor) agonists and antagonists

Cited by 61 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. The multicomponent Passerini reaction as a means of accessing diversity in structure, activity and properties: Soft and hard vanilloid/cannabinoid modulators;European Journal of Medicinal Chemistry;2024-12

2. Three-Step Synthesis of N-(7-chloro-4-morpholinoquinolin-2-yl)benzamide from 4,7-Dichloroquinoline;Molbank;2024-03-21

3. Capsaicin derivatives: Synthesis and biological activity;Chemical Biology & Drug Design;2024-02

4. The Multicomponent Passerini Reaction as a Means of Accessing Diversity in Structure, Activity and Properties: Soft and Hard Vanilloid/Cannabinoid Modulators;2024

5. Non-Canonical Cannabinoid Receptors with Distinct Binding and Signaling Properties in Prostate and Other Cancer Cell Types Mediate Cell Death;International Journal of Molecular Sciences;2022-03-11