Stereospecific, Stereoselective Rearrangement of Hexahydro-1,3-diazepin-2-ones to Tetrahydropyrimidin-2-ones and Imidazolidin-2-ones, a Useful Route for the Synthesis of HIV Protease Inhibitors-Reference-Cited by-同舟云学术

Stereospecific, Stereoselective Rearrangement of Hexahydro-1,3-diazepin-2-ones to Tetrahydropyrimidin-2-ones and Imidazolidin-2-ones, a Useful Route for the Synthesis of HIV Protease Inhibitors

Published:1998-06-20 Issue:14 Volume:63 Page:4755-4766
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

De Lucca George V.¹

Affiliation:

1. Dupont Merck Pharmaceutical Company, Wilmington, Delaware 19880-0500

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo980533e

Reference19 articles.

1. L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor.

2. ABT-538 is a potent inhibitor of human immunodeficiency virus protease and has high oral bioavailability in humans.

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