Predicting Intrinsic Aqueous Solubility by a Thermodynamic Cycle-Reference-Cited by-同舟云学术

Predicting Intrinsic Aqueous Solubility by a Thermodynamic Cycle

Published:2008-02-22 Issue:2 Volume:5 Page:266-279
ISSN:1543-8384
Container-title:Molecular Pharmaceutics
language:en
Short-container-title:Mol. Pharmaceutics

Author:

Palmer David S.¹,Llinàs Antonio¹,Morao Iñaki¹,Day Graeme M.¹,Goodman Jonathan M.¹,Glen Robert C.¹,Mitchell John B. O.¹

Affiliation:

1. The Pfizer Institute for Pharmaceutical Materials Science and Unilever Centre for Molecular Science Informatics, Department of Chemistry, University of Cambridge, Lensfield Road, Cambridge, CB2 1EW, United Kingdom, and Pfizer Global Research and Development, Sandwich Laboratories, Sandwich, Kent CT13 9NJ, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/mp7000878

Reference72 articles.

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2. Yalkowsky, S. H.Solubility and Solubilization in Aqueous Media;Oxford University Press:New York, 1999; p67.

3. THE RATE OF SOLUTION OF SOLID SUBSTANCES IN THEIR OWN SOLUTIONS.

4. Relationship Between In Vitro Dissolution Rates and Solubilities of Numerous Compounds Representative of Various Chemical Species

5. In vitro models for processes involved in intestinal absorption

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