Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine Derivatives as Adenosine Receptor Antagonists. Influence of the N5 Substituent on the Affinity at the Human A3 and A2B Adenosine Receptor Subtypes: A Molecular Modeling Investigation-Reference-Cited by-同舟云学术

Pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine Derivatives as Adenosine Receptor Antagonists. Influence of the N5 Substituent on the Affinity at the Human A3 and A2B Adenosine Receptor Subtypes: A Molecular Modeling Investigation

Published:2003-08-30 Issue:20 Volume:46 Page:4287-4296
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pastorin Giorgia¹,Da Ros Tatiana¹,Spalluto Giampiero¹,Deflorian Francesca¹,Moro Stefano¹,Cacciari Barbara¹,Baraldi Pier Giovanni¹,Gessi Stefania¹,Varani Katia¹,Borea Pier Andrea¹

Affiliation:

1. Dipartimento di Scienze Farmaceutiche, Università degli Studi di Trieste, Piazzale Europa 1, I-34127 Trieste, Italy, Dipartimento di Scienze Farmaceutiche, Università degli Studi di Ferrara, Via Fossato di Mortara 17-19, I-44100 Ferrara, Italy, Molecular Modeling Section, Dipartimento di Scienze Farmaceutiche, Università di Padova, via Marzolo 5, I-35131 Padova, Italy, and Dipartimento di Medicina Clinica e Sperimentale-Sezione di Farmacologia, Università degli Studi di Ferrara, Via Fossato di Mortara 17...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030852k

Reference46 articles.

1. A3 Adenosine Receptor Ligands: History and Perspectives

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