Development of Inhibitors of the PAS-B Domain of the HIF-2α Transcription Factor-Reference-Cited by-同舟云学术

Development of Inhibitors of the PAS-B Domain of the HIF-2α Transcription Factor

Published:2013-02-18 Issue:4 Volume:56 Page:1739-1747
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rogers Jamie L.¹,Bayeh Liela¹,Scheuermann Thomas H.¹,Longgood Jamie¹,Key Jason¹,Naidoo Jacinth¹,Melito Lisa¹,Shokri Cameron¹,Frantz Doug E.¹,Bruick Richard K.¹,Gardner Kevin H.¹,MacMillan John B.¹,Tambar Uttam K.¹

Affiliation:

1. Departments of Biochemistry and Biophysics, University of Texas Southwestern Medical Center, 5323 Harry Hines Boulevard, Dallas, Texas 75390-9038, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm301847z

Reference30 articles.

1. Hypoxia-inducible factors: mediators of cancer progression and targets for cancer therapy

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3. High-resolution genome-wide mapping of HIF-binding sites by ChIP-seq

4. Levels of hypoxia-inducible factor-1? independently predict prognosis in patients with lymph node negative breast carcinoma

5. Expression of hypoxia-inducible factor 1? in brain tumors

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