A Nonionic Inhibitor with High Specificity for the UDP-Gal Donor Binding Site of Human Blood Group B Galactosyltransferase: Design, Synthesis, and Characterization-Reference-Cited by-同舟云学术

A Nonionic Inhibitor with High Specificity for the UDP-Gal Donor Binding Site of Human Blood Group B Galactosyltransferase: Design, Synthesis, and Characterization

Published:2013-02-28 Issue:5 Volume:56 Page:2150-2154
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Schaefer Katrin¹,Sindhuwinata Nora²,Hackl Thomas¹,Kötzler Miriam P.¹,Niemeyer Felix C.¹,Palcic Monica M.³,Peters Thomas²,Meyer Bernd¹

Affiliation:

1. Organic Chemistry, Department of Chemistry, Faculty of Sciences, University of Hamburg, Martin Luther King Platz 6, 20146 Hamburg, Germany

2. Institute of Chemistry, University of Luebeck, Ratzeburger Allee 160, 23538 Luebeck, Germany

3. Carlsberg Laboratory, Gamle Carlsberg Vej 10, 1799 Copenhagen V, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300642a

Reference30 articles.

1. Glycosyltransferases: Structures, Functions, and Mechanisms

2. Carbohydrate mimetics-based glycosyltransferase inhibitors

3. Bisubstrate Analogues as Glycosyltransferase Inhibitors

4. Synthesis of Glycosyltransferase Inhibitors

5. Antigen structure and genetic basis of histo-blood groups A, B and O: their changes associated with human cancer

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