Chiral 1,3,4-Oxadiazol-2-ones as Highly Selective FAAH Inhibitors

Author:

Patel Jayendra Z.1,Parkkari Teija12,Laitinen Tuomo1,Kaczor Agnieszka A.13,Saario Susanna M.2,Savinainen Juha R.2,Navia-Paldanius Dina2,Cipriano Mariateresa4,Leppänen Jukka1,Koshevoy Igor O.5,Poso Antti1,Fowler Christopher J.4,Laitinen Jarmo T.2,Nevalainen Tapio1

Affiliation:

1. School of Pharmacy, Faculty of Health Sciences, University of Eastern Finland, P.O. Box 1627, FIN-70211 Kuopio, Finland

2. School of Medicine, Institute of Biomedicine/Physiology, University of Eastern Finland, P.O. Box 1627, FIN-70211 Kuopio, Finland

3. Department of Synthesis and Chemical Technology of Pharmaceutical Substances, Faculty of Pharmacy with Division of Medical Analytics, Medical University of Lublin, 4a Chodzki Street, PL-20093 Lublin, Poland

4. Department of Pharmacology and Clinical Neuroscience, Umeå University, SE-90187, Umeå, Sweden

5. Department of Chemistry, University of Eastern Finland, P.O. Box 111, FIN-80101 Joensuu, Finland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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