Identification of Potent and Selective Non-covalent Inhibitors of the Plasmodium falciparum Proteasome
Author:
Affiliation:
1. Takeda Pharmaceuticals International Co., 40 Landsdowne Street, Cambridge, Massachusetts 02139, United States
Funder
Agency for Science, Technology and Research
National Institute of Allergy and Infectious Diseases
Publisher
American Chemical Society (ACS)
Subject
Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis
Link
https://pubs.acs.org/doi/pdf/10.1021/ja507692y
Reference18 articles.
1. World Health Organization, World Malaria Report 2013.
2. Evolutionary origin of Plasmodium and other Apicomplexa based on rRNA genes.
3. Assembly, structure, and function of the 26S proteasome
4. Proteasome Inhibitors: An Expanding Army Attacking a Unique Target
Cited by 48 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Emerging Drug Targets for Antimalarial Drug Discovery: Validation and Insights into Molecular Mechanisms of Function;Journal of Medicinal Chemistry;2024-01-10
2. Identification of new drug candidates against Trichomonas gallinae using high-throughput screening;International Journal for Parasitology: Drugs and Drug Resistance;2023-12
3. Covalent Macrocyclic Proteasome Inhibitors Mitigate Resistance in Plasmodium falciparum;ACS Infectious Diseases;2023-09-15
4. Covalent macrocyclic proteasome inhibitors mitigate resistance inPlasmodium falciparum;2023-07-03
5. Dual-pharmacophore artezomibs hijack the Plasmodium ubiquitin-proteasome system to kill malaria parasites while overcoming drug resistance;Cell Chemical Biology;2023-05
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3