Selective CRAF Inhibition Elicits Transactivation-Reference-Cited by-同舟云学术

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Selective CRAF Inhibition Elicits Transactivation

Published:2021-03-22 Issue:12 Volume:143 Page:4600-4606
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Morgan Charles W.¹^ORCID,Dale Ian L.²,Thomas Andrew P.³,Hunt James⁴,Chin Jason W.¹^ORCID

Affiliation:

1. Medical Research Council Laboratory of Molecular Biology, Cambridge CB2 0QH, United Kingdom

2. Discovery Sciences, R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom

3. Medicinal Chemistry, Oncology R&D, AstraZeneca, Cambridge CB4 0WG, United Kingdom

4. Antibody Discovery & Protein Engineering, R&D, AstraZeneca, Cambridge CB21 6GH, United Kingdom

Funder

Medical Research Council

AstraZeneca UK Limited

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/jacs.0c11958

Reference67 articles.

1. Unnatural Ligands for Engineered Proteins: New Tools for Chemical Genetics

2. A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes

3. Bump-and-Hole Engineering Identifies Specific Substrates of Glycosyltransferases in Living Cells

4. Design of Allele-Specific Protein Methyltransferase Inhibitors

5. Proteome labeling and protein identification in specific tissues and at specific developmental stages in an animal

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1. Engineering Pyrrolysine Systems for Genetic Code Expansion and Reprogramming;Chemical Reviews;2024-09-05

2. Targeting RAF dimers in RAS mutant tumors: From biology to clinic;Acta Pharmaceutica Sinica B;2024-05

3. The Pan-RAF–MEK Nondegrading Molecular Glue NST-628 Is a Potent and Brain-Penetrant Inhibitor of the RAS–MAPK Pathway with Activity across Diverse RAS- and RAF-Driven Cancers;Cancer Discovery;2024-04-19

4. 14-3-3 interaction with phosphodiesterase 8A sustains PKA signaling and downregulates the MAPK pathway;Journal of Biological Chemistry;2024-03

5. Targeting CRAF kinase in anti-cancer therapy: progress and opportunities;Molecular Cancer;2023-12-18

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