A New Pyridazine Series of GABAA α5 Ligands-Reference-Cited by-同舟云学术

A New Pyridazine Series of GABAA α5 Ligands

Published:2005-08-23 Issue:19 Volume:48 Page:6004-6011
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

van Niel Monique B.¹,Wilson Kevin¹,Adkins Charles H.¹,Atack John R.¹,Castro José L.¹,Clarke Dawn E.¹,Fletcher Stephen¹,Gerhard Ute¹,Mackey Mark M.¹,Malpas Sallie¹,Maubach Karen¹,Newman Robert¹,O'Connor Desmond¹,Pillai Gopalan V.¹,Simpson Peter B.¹,Thomas Steven R.¹,MacLeod Angus M.¹

Affiliation:

1. Departments of Medicinal Chemistry, Biochemistry and Pharmacology, Merck Sharp & Dohme Research Laboratories, Terlings Park, Eastwick Road, Harlow, Essex, CM20 2QR, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm050249x

Reference28 articles.

1. The neuropharmacological and neurochemical basis of place learning in the Morris water maze

2. The GABA-A receptor gene family: new targets for therapeutic intervention

3. Importance of a novel GABAA receptor subunit for benzodiazepine pharmacology

4. The distribution of 13 GABAA receptor subunit mRNAs in the rat brain. I. Telencephalon, diencephalon, mesencephalon

5. Enhanced Learning and Memory and Altered GABAergic Synaptic Transmission in Mice Lacking the α5 Subunit of the GABAAReceptor

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