Complementarity between in Silico and Biophysical Screening Approaches in Fragment-Based Lead Discovery against the A2A Adenosine Receptor
Author:
Affiliation:
1. ZoBio BV, 2300RA Leiden, The Netherlands
2. Science for Life Laboratory, SE-171 21 Solna, Sweden
3. Department of Biochemistry and Biophysics and Center for Biomembrane Research, Stockholm University, SE-106 91 Stockholm, Sweden
Publisher
American Chemical Society (ACS)
Subject
Library and Information Sciences,Computer Science Applications,General Chemical Engineering,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/ci4003156
Reference79 articles.
1. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update
2. Adenosine Receptors and Inflammation
3. Adenosine Receptors and the Central Nervous System
4. Diversity and modularity of G protein-coupled receptor structures
5. Progress in Structure Based Drug Design for G Protein-Coupled Receptors
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