Bicyclo[2.2.1]heptane and 6,6-Dimethylbicyclo[3.1.1]heptane Derivatives: Orally Active, Potent, and Selective Prostaglandin D2 Receptor Antagonists-Reference-Cited by-同舟云学术

Bicyclo[2.2.1]heptane and 6,6-Dimethylbicyclo[3.1.1]heptane Derivatives: Orally Active, Potent, and Selective Prostaglandin D2 Receptor Antagonists

Published:1997-10-01 Issue:22 Volume:40 Page:3504-3507
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Tsuri Tatsuo¹,Honma Tsunetoshi¹,Hiramatsu Yoshiharu¹,Okada Toshihiko¹,Hashizume Hiroshi¹,Mitsumori Susumu¹,Inagaki Masanao¹,Arimura Akinori¹,Yasui Kiyoshi¹,Asanuma Fujio¹,Kishino Junji¹,Ohtani Mitsuaki¹

Affiliation:

1. Shionogi Research Laboratories, Shionogi & Co., Ltd., Fukushima-ku, Osaka 553, Japan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970343g

Reference37 articles.

1. INFLAMMATORY EFFECTS OF PROSTAGLANDIN D2 IN RAT AND HUMAN SKIN

2. Physiologic responses to intranasal dose-response challenges with histamine, methacholine, bradykinin, and prostaglandin in adult volunteers with and without nasal allergy

3. Prostaglandin D₂-induced bronchoconstriction is mediated only in part by the thromboxane prostanoid receptor

Cited by 37 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis of bridged tricyclo[5.2.1.01,5]decanes via nickel-catalyzed asymmetric domino cyclization of enynones;Nature Communications;2020-04-20

2. Effect of the potent and selective DP1 receptor antagonist, asapiprant (S-555739), in animal models of allergic rhinitis and allergic asthma;European Journal of Pharmacology;2015-10

3. Discovery of selective indole-based prostaglandin D2 receptor antagonist;Bioorganic & Medicinal Chemistry;2011-08

4. Prostaglandins and Inflammation;Arteriosclerosis, Thrombosis, and Vascular Biology;2011-05

5. Understanding DP receptor antagonism using a CoMSIA approach;Bioorganic & Medicinal Chemistry Letters;2011-01