Inhibitors of Multiple Mutants of Plasmodium falciparum Dihydrofolate Reductase and Their Antimalarial Activities-Reference-Cited by-同舟云学术

Inhibitors of Multiple Mutants of Plasmodium falciparum Dihydrofolate Reductase and Their Antimalarial Activities

Published:2003-12-23 Issue:3 Volume:47 Page:673-680
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kamchonwongpaisan Sumalee¹,Quarrell Rachel¹,Charoensetakul Netnapa¹,Ponsinet Rachel¹,Vilaivan Tirayut¹,Vanichtanankul Jarunee¹,Tarnchompoo Bongkoch¹,Sirawaraporn Worachart¹,Lowe Gordon¹,Yuthavong Yongyuth¹

Affiliation:

1. National Center for Genetic Engineering and Biotechnology, National Science and Technology Development Agency, Pathumthani 12120, Thailand; Department of Chemistry, Faculty of Science, Chulalongkorn University, Bangkok 10330, Thailand; Department of Biochemistry, Faculty of Science, Mahidol University, Bangkok 10400, Thailand, and The Dyson Perrins Laboratory, Department of Chemistry, Oxford University, South Parks Road, Oxford, OX1 3QY, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030165t

Reference22 articles.

1. Basis for antifolate action and resistance in malaria

2. Resistance to antifolates in Plasmodium falciparum monitored by sequence analysis of dihydropteroate synthetase and dihydrofolate reductase alleles in a large number of field samples of diverse origins

3. P. falciparum dihydrofolate reductase and dihydropteroate synthase mutations: epidemiology and role in clinical resistance to antifolates

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