Molecular Determinants of Ligand Binding Modes in the Histamine H4 Receptor: Linking Ligand-Based Three-Dimensional Quantitative Structure–Activity Relationship (3D-QSAR) Models to in Silico Guided Receptor Mutagenesis Studies-Reference-Cited by-同舟云学术

Molecular Determinants of Ligand Binding Modes in the Histamine H4 Receptor: Linking Ligand-Based Three-Dimensional Quantitative Structure–Activity Relationship (3D-QSAR) Models to in Silico Guided Receptor Mutagenesis Studies

Published:2011-11-07 Issue:23 Volume:54 Page:8136-8147
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Istyastono Enade P.¹,Nijmeijer Saskia¹,Lim Herman D.²,van de Stolpe Andrea¹,Roumen Luc¹,Kooistra Albert J.¹,Vischer Henry F.¹,de Esch Iwan J. P.¹,Leurs Rob¹,de Graaf Chris¹

Affiliation:

1. Department of Pharmacochemistry, Faculty of Exact Sciences, Leiden/Amsterdam Center for Drug Research (LACDR), Division of Medicinal Chemistry, VU University Amsterdam, De Boelelaan 1083, 1081 HV Amsterdam, The Netherlands

2. Department of Medicinal Chemistry, Room P-246, Griffin Discoveries BV, De Boelelaan 1083, 1081 HV, Amsterdam, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201042n

Reference61 articles.

1. Molecular Determinants of Selective Agonist and Antagonist Binding to the Histamine H4 Receptor

2. Cloning and Pharmacological Characterization of a Fourth Histamine Receptor (H4) Expressed in Bone Marrow

3. Major advances in the development of histamine H4 receptor ligands

4. The role of histamine H1 and H4 receptors in allergic inflammation: the search for new antihistamines

5. The role of histamine H4 receptor in immune and inflammatory disorders

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