Highly Potent, Selective, and Orally Active Phosphodiesterase 10A Inhibitors-Reference-Cited by-同舟云学术

Highly Potent, Selective, and Orally Active Phosphodiesterase 10A Inhibitors

Published:2011-10-11 Issue:21 Volume:54 Page:7621-7638
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Malamas Michael S.¹,Ni Yike¹,Erdei James¹,Stange Hans²,Schindler Rudolf²,Lankau Hans-Joachim²,Grunwald Christian²,Fan Kristi Yi¹,Parris Kevin¹,Langen Barbara²,Egerland Ute²,Hage Thorsten²,Marquis Karen L.¹,Grauer Steve¹,Brennan Julie¹,Navarra Rachel¹,Graf Radka¹,Harrison Boyd L.¹,Robichaud Albert¹,Kronbach Thomas²,Pangalos Menelas N.¹,Hoefgen Norbert²,Brandon Nicholas J.³

Affiliation:

1. Pfizer Neuroscience Princeton, 865 Ridge Road, Monmouth Junction, New Jersey 08852, United States

2. Biocrea Therapies GmbH, Meissner Strasse 191, 01445 Radebeul, Germany

3. Pfizer Neuroscience, Eastern Point Road, Groton Connecticut 06340, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm2009138

Reference22 articles.

1. The Next Generation of Phosphodiesterase Inhibitors: Structural Clues to Ligand and Substrate Selectivity of Phosphodiesterases

2. Inhibitors of PDE4: a review of recent patent literature

3. Phosphodiesterase 5 inhibitors: current status and potential applications

4. Keynote review: Phosphodiesterase-4 as a therapeutic target

5. Cyclic Nucleotide Phosphodiesterases: Molecular Regulation to Clinical Use

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