Ortho Lithiation of N-Pivaloylfluoroanilines as a Useful Tool for Either Selective Methylation or Benzoxazole Synthesis-Reference-Cited by-同舟云学术

Ortho Lithiation of N-Pivaloylfluoroanilines as a Useful Tool for Either Selective Methylation or Benzoxazole Synthesis

Published:2004-10-29 Issue:6 Volume:8 Page:958-961
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Yoshida Yasuo¹,Hamada Yusuke¹,Umezu Kazuto¹,Tabuchi Fumiya¹

Affiliation:

1. Research and Development Department, Ihara Chemical Industry Co., Ltd., Fujikawa-cho, Ihara-gun, Shizuoka 421-3306, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op0498969

Reference10 articles.

1. A novel synthesis of the intermediate which can be useful for antimicrobacterial agent such as HSR-903 is described; see: Hamada, Y.; Umezu, K. Patent Application No. JP11-035531.

2. Hamada, Y.; Umezu, K. Patent Application No. JP11-158150.

3. Directed ortho metalation. Tertiary amide and O-carbamate directors in synthetic strategies for polysubstituted aromatics

4. A practical route to C-8 substituted fluoroquinolones

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