Synthesis and Anti-HIV Activity of Cosalane Analogues with Substituted Benzoic Acid Rings Attached to the Pharmacophore through Methylene and Amide Linkers-Reference-Cited by-同舟云学术

Synthesis and Anti-HIV Activity of Cosalane Analogues with Substituted Benzoic Acid Rings Attached to the Pharmacophore through Methylene and Amide Linkers

Published:1999-07-14 Issue:16 Volume:64 Page:5858-5866
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Ruell Jeffrey A.¹,De Clercq Erik¹,Pannecouque Christophe¹,Witvrouw Myriam¹,Stup Tracy L.¹,Turpin Jim A.¹,Buckheit, Robert W.¹,Cushman Mark¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, School of Pharmacy and Pharmacal Sciences, Purdue University, West Lafayette, Indiana 47907, Rega Institute for Medical Research, Katholieke Universiteit Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium, and Virology Research Group, Serquest, 431 Aviation Way, Frederick, Maryland 21701

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo990177f

Reference24 articles.

1. Design and synthesis of cosalane, a novel anti-HIV agent

2. Lipophilic bis-arylsulfonates as inhibitors of the CD4-gp120 interaction

3. Correlation of Anti-HIV Potency with Lipophilicity in a Series of Cosalane Analogs Having Normal Alkenyl and Phosphodiester Chains as Cholestane Replacements

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