Bicyclic Picomolar OGA Inhibitors Enable Chemoproteomic Mapping of Its Endogenous Post-translational Modifications

Author:

González-Cuesta Manuel1ORCID,Sidhu Peter23,Ashmus Roger A.2ORCID,Males Alexandra4,Proceviat Cameron2,Madden Zarina2,Rogalski Jason C.3,Busmann Jil A.5,Foster Leonard J.3,García Fernández José M.6ORCID,Davies Gideon J.4ORCID,Ortiz Mellet Carmen1ORCID,Vocadlo David J.25ORCID

Affiliation:

1. Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, 41012 Sevilla, Spain

2. Department of Chemistry, Simon Fraser University, Burnaby, British Columbia V5A 1S6, Canada

3. Department of Biochemistry and Molecular Biology, University of British Columbia, Vancouver, British Columbia V6T 1Z4, Canada

4. Department of Chemistry. University of York, York YO10 5DD, United Kingdom

5. Department of Molecular Biology and Biochemistry, Simon Fraser University, Burnaby, British Columbia V5A 1S6, Canada

6. Instituto de Investigaciones Químicas (IIQ), CSIC, Universidad de Sevilla, 41092 Sevilla, Spain

Funder

Canadian Institutes of Health Research

Junta de Andaluc?a

Canada Foundation for Innovation

Ministerio de Ciencia e Innovaci?n

European Regional Development Fund

Canada Research Chairs

Genome Canada

British Columbia Knowledge Development Fund

Michael Smith Foundation for Health Research

Agencia Estatal de Investigaci?n, Ministerio de Ciencia, Innovaci?n y Universidades

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

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