A Modular and Diastereoselective 5 + 1 Cyclization Approach to N-(Hetero)Aryl Piperidines-Reference-Cited by-同舟云学术

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A Modular and Diastereoselective 5 + 1 Cyclization Approach to N-(Hetero)Aryl Piperidines

Published:2019-12-27 Issue:2 Volume:142 Page:726-732
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Larsen Matthew A.¹^ORCID,Hennessy Elisabeth T.¹,Deem Madeleine C.²,Lam Yu-hong³^ORCID,Saurí Josep⁴,Sather Aaron C.²^ORCID

Affiliation:

1. Department of Discovery Chemistry, Merck & Co., Inc., Boston, Massachusetts 02115, United States

2. Department of Process Research and Development, Merck & Co., Inc., Boston, Massachusetts 02115, United States

3. Computational and Structural Chemistry, Merck & Co., Inc., P.O. Box 2000, Rahway, New Jersey 07065, United States

4. Analytical Research and Development, Merck & Co., Inc., Boston, Massachusetts 02115, United States

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/jacs.9b13114

Reference46 articles.

1. Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

2. Rings in Drugs

3. Recent contributions from the asymmetric aza-Michael reaction to alkaloids total synthesis

4. Stereocontrolled synthesis of vicinally functionalized piperidines by nucleophilic β-addition of alkyllithiums to α-aryl substituted piperidine enecarbamates

5. Enantioselective Synthesis of Chiral Piperidines via the Stepwise Dearomatization/Borylation of Pyridines

Cited by 21 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Regio‐ and Diastereoselective Synthesis of Polysubstituted Piperidines Enabled by Boronyl Radical‐Catalyzed (4+2) Cycloaddition;Angewandte Chemie International Edition;2024-08-19

2. Regio‐ and Diastereoselective Synthesis of Polysubstituted Piperidines Enabled by Boronyl Radical‐Catalyzed (4+2) Cycloaddition;Angewandte Chemie;2024-08-19

3. Discovery Process Chemistry: An Innovation Hub at the Interface of Academia, the Pharmaceutical Industry, and Contract Research Organization;Synthesis;2024-08-05

4. Reductive Transamination of Pyridinium Salts to N-Aryl Piperidines;The Journal of Organic Chemistry;2024-06-13

5. Palladium-Catalyzed Allylation of Endocyclic 1-Azaallyl Anions;The Journal of Organic Chemistry;2024-06-10

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