Design, Synthesis, and in Vitro Pharmacology of New Radiolabeled γ-Hydroxybutyric Acid Analogues Including Photolabile Analogues with Irreversible Binding to the High-Affinity γ-Hydroxybutyric Acid Binding Sites-Reference-Cited by-同舟云学术

Design, Synthesis, and in Vitro Pharmacology of New Radiolabeled γ-Hydroxybutyric Acid Analogues Including Photolabile Analogues with Irreversible Binding to the High-Affinity γ-Hydroxybutyric Acid Binding Sites

Published:2010-08-17 Issue:17 Volume:53 Page:6506-6510
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Sabbatini Paola¹,Wellendorph Petrine¹,Høg Signe¹,Pedersen Martin H. F.²,Bräuner-Osborne Hans¹,Martiny Lars²,Frølund Bente¹,Clausen Rasmus P.¹

Affiliation:

1. Department of Medicinal Chemistry, Faculty of Pharmaceutical Sciences, University of Copenhagen, 2 Universitetsparken, Dk-2100 Copenhagen, Denmark

2. The Hevesy Laboratory, Radiation Research Division, Risø, The Technical University of Denmark, 399 Frederiksborgvej, Dk-4000 Roskilde, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm1006325

Reference25 articles.

1. Gamma-Hydroxybutyrate, a Normal Brain Metabolite

2. THE γ-HYDROXYBUTYRATE SIGNALLING SYSTEM IN BRAIN: ORGANIZATION AND FUNCTIONAL IMPLICATIONS

3. Sodium Oxybate

4. Gamma Hydroxybutyric Acid (GHB) for the Treatment of Alcohol Dependence: A Review

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