Potent N-(1,3-Thiazol-2-yl)pyridin-2-amine Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors with Excellent Pharmacokinetics and Low Affinity for the hERG Ion Channel
Author:
Affiliation:
1. Departments of Medicinal Chemistry, Cancer Research, Drug Metabolism and Pharmacology, Merck Research Laboratories, P.O. Box 4, West Point, Pennsylvania 19486
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm049697f
Reference23 articles.
1. The Biology of Vascular Endothelial Growth Factor
2. Vascular endothelial growth factor (VEGF) and its receptors
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