Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups-Reference-Cited by-同舟云学术

Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups

Published:2014-10-17 Issue:21 Volume:57 Page:9152-9167
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bozdag Murat¹,Ferraroni Marta¹,Carta Fabrizio¹,Vullo Daniela¹,Lucarini Laura²,Orlandini Elisabetta³,Rossello Armando³,Nuti Elisa³,Scozzafava Andrea¹,Masini Emanuela²,Supuran Claudiu T.¹⁴

Affiliation:

1. Laboratorio di Chimica Bioinorganica, Polo Scientifico, Università degli Studi di Firenze, Rm. 188, Via della Lastruccia 3, 50019 Sesto Fiorentino, Florence, Italy

2. Sezione di Farmacologia, Dipartimento di Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA), Università degli Studi di Firenze, Viale Pieraccini 6, 50139 Florence, Italy

3. Dipartimento di Farmacia, Università di Pisa, Via Bonanno, 6, 56126 Pisa, Italy

4. Sezione di Scienze Farmaceutiche, Dipartimento di Neuroscienze, Psicologia, Area del Farmaco e Salute del Bambino (NEUROFARBA), Università degli Studi di Firenze, Via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy

Funder

European Commission

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501314c

Reference79 articles.

1. Evolution of a new enzyme for carbon disulphide conversion by an acidothermophilic archaeon

2. Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?

3. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators