Synthesis and Anticonvulsant Activity of Novel and Potent 2,3-Benzodiazepine AMPA/Kainate Receptor Antagonists-Reference-Cited by-同舟云学术

Synthesis and Anticonvulsant Activity of Novel and Potent 2,3-Benzodiazepine AMPA/Kainate Receptor Antagonists

Published:1999-09-23 Issue:21 Volume:42 Page:4414-4421
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Grasso Silvana¹,De Sarro Giovambattista¹,De Sarro Angela¹,Micale Nicola¹,Zappalà Maria¹,Puia Giulia¹,Baraldi Mario¹,De Micheli Carlo¹

Affiliation:

1. Dipartimento Farmaco-Chimico and Istituto di Farmacologia, Università di Messina, Italy, Dipartimento di Medicina Sperimentale e Clinica, Università di Catanzaro, Italy, Dipartimento di Scienze Farmaceutiche, Università di Modena, Italy, and Istituto di Chimica Farmaceutica, Università di Milano, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm991086d

Reference36 articles.

1. GYKI 52466, a 2,3-benzodiazepine, is a highly selective, noncompetitive antagonist of AMPA/kainate receptor responses

2. Therapeutic potential of excitatory amino acid antagonists: channel blockers and 2,3-benzodiazepines

3. The anticonvulsant effect of the non-NMDA antagonists, NBQX and GYKI 52466, in mice

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