Synthesis of New Steroidal Inhibitors of P-Glycoprotein-Mediated Multidrug Resistance and Biological Evaluation on K562/R7 Erythroleukemia Cells-Reference-Cited by-同舟云学术

Synthesis of New Steroidal Inhibitors of P-Glycoprotein-Mediated Multidrug Resistance and Biological Evaluation on K562/R7 Erythroleukemia Cells

Published:2015-02-11 Issue:4 Volume:58 Page:1832-1845
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

de Ravel Marc Rolland¹²,Alameh Ghina²,Melikian Maxime²,Mahiout Zahia²,Emptoz-Bonneton Agnès²,Matera Eva-Laure¹,Lomberget Thierry²³,Barret Roland²³,Rocheblave Luc²³,Walchshofer Nadia²³,Beltran Sonia²,El Jawad Lucienne²,Mappus Elisabeth²,Grenot Catherine²,Pugeat Michel³,Dumontet Charles¹,Le Borgne Marc²³,Cuilleron Claude Yves²

Affiliation:

1. Centre de Recherche en Cancérologie de Lyon - Université Claude Bernard Lyon 1, INSERM U1052-CNRS UMR5286, Centre Léon Bérard-Cheney D, 28 rue Laënnec, Lyon 69373 Cedex 08, France

2. INSERM-U863 Hormones stéroïdes et protéines de liaison, Université Claude Bernard Lyon 1, 8 Avenue Rockefeller, Lyon 69373 Cedex 08, France

3. Université de Lyon, Université Claude Bernard Lyon 1, Faculté de Pharmacie, ISPB, EA 4446 Biomolécules Cancer et Chimiorésistances, SFR Santé Lyon-Est CNRS UMS3453-INSERM US7, 8 Avenue Rockefeller, Lyon 69373 Cedex 08 France

Funder

Institut national de la santé et de la recherche médicale

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm501676v

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