Allosteric Antagonist Modulation of TRPV2 by Piperlongumine Impairs Glioblastoma Progression

Author:

Conde João1ORCID,Pumroy Ruth A.2,Baker Charlotte1,Rodrigues Tiago1,Guerreiro Ana1,Sousa Bárbara B.1,Marques Marta C.1,de Almeida Bernardo P.1,Lee Sohyon3,Leites Elvira P.1,Picard Daniel456,Samanta Amrita2,Vaz Sandra H.1ORCID,Sieglitz Florian1,Langini Maike456,Remke Marc456,Roque Rafael7,Weiss Tobias8,Weller Michael8,Liu Yuhang9,Han Seungil9,Corzana Francisco10ORCID,Morais Vanessa A.1,Faria Cláudia C.111,Carvalho Tânia1,Filippakopoulos Panagis12,Snijder Berend3,Barbosa-Morais Nuno L.1,Moiseenkova-Bell Vera Y.2,Bernardes Gonçalo J. L.113ORCID

Affiliation:

1. Instituto de Medicina Molecular João Lobo Antunes, Faculdade de Medicina, Universidade de Lisboa, Av. Prof. Egas Moniz, 1649-028 Lisboa, Portugal

2. Department of Systems Pharmacology and Translational Therapeutics, Perelman School of Medicine, University of Pennsylvania, Philadelphia, Pennsylvania 19104, United States

3. Institute of Molecular Systems Biology, ETH Zürich, Otto-Stern-Weg 3, 8093 Zürich, Switzerland

4. Department of Pediatric Neuro-Oncogenomics, DKFZ, Heidelberg 69120, Germany

5. Department of Pediatric Neuro-Oncogenomics, DKTK, Essen D-45147, Germany

6. Department of Pediatric Oncology, Hematology, and Clinical Immunology, Medical Faculty, University Hospital Düsseldorf, Düsseldorf 40225, Germany

7. Laboratório de Neuropatologia, Hospital de Santa Maria, Centro Hospitalar Universitário Lisboa Norte (CHLN) EPE, Av. Prof. Egas Moniz, 1649-028 Lisboa, Portugal

8. Department of Neurology and Brain Tumour Center, University Hospital Zürich and University of Zurich, Rämistrasse 100, 8091 Zürich, Switzerland

9. Discovery Sciences, Worldwide Research and Development, Pfizer Inc., Eastern Point Road, Groton, Connecticut 06340, United States

10. Departamento de Química, Universidad de La Rioja, 26006 Logroño, Spain

11. Department of Neurosurgery, Hospital de Santa Maria, Centro Hospitalar Universitário Lisboa Norte (CHULN) EPE, Av. Prof. Egas Moniz, 1649-028 Lisboa, Portugal

12. Structural Genomics Consortium, Oxford University, Old Road Campus Research Building, Roosevelt Drive, OX3 7DQ Oxford, United Kingdom

13. Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, CB2 1EW Cambridge, United Kingdom

Funder

Royal Society

Medical Research Council

Horizon 2020 Framework Programme

National Institutes of Health

Funda??o para a Ci?ncia e a Tecnologia

European Molecular Biology Organization

Agencia Estatal Investigaci?n of Spain

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

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