An Atom-Economical Method To Prepare Enantiopure Benzodiazepines with N-Carboxyanhydrides
Author:
Affiliation:
1. Department of Process Research and Development, Merck & Co., Inc., Rahway, New Jersey 07065, United States
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.7b00417
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3. Facile and Efficient One‐Pot Protocol for Synthesis of 5‐Phenyl‐1,4‐benzodiazepine‐2‐one Derivatives
4. Enantioselective Synthesis of Diversely Substituted Quaternary 1,4-Benzodiazepin-2-ones and 1,4-Benzodiazepine-2,5-diones
5. Diastereoselective Pictet−Spengler Approach for the Synthesis of Pyrrolo[3,2-e][1,4]diazepin-2-one Peptide Turn Mimics
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