Direct Synthesis of 3-Acylindoles through Rhodium(III)-Catalyzed Annulation of N-Phenylamidines with α-Cl Ketones-Reference-Cited by-同舟云学术

Direct Synthesis of 3-Acylindoles through Rhodium(III)-Catalyzed Annulation of N-Phenylamidines with α-Cl Ketones

Published:2018-11-20 Issue:23 Volume:20 Page:7645-7649
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Zhou Jianhui¹,Li Jian²,Li Yazhou²,Wu Chenglin²,He Guoxue²,Yang Qiaolan²,Zhou Yu²^ORCID,Liu Hong²^ORCID

Affiliation:

1. School of Pharmacy, Nanchang University, 461 Bayi Road, Nanchang 330006, China

2. State Key Laboratory of Drug Research and Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zu Chong Zhi Road, Shanghai 201203, China

Funder

National Natural Science Foundation of China

Chinese Academy of Sciences

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.8b03383

Reference47 articles.

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2. Simple indole alkaloids and those with a nonrearranged monoterpenoid unit

3. Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety

4. Conformationally restrained analogs of pravadoline: nanomolar potent, enantioselective, (aminoalkyl)indole agonists of the cannabinoid receptor

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