Rhodium(III)-Catalyzed C–H Activation: Ligand-Controlled Regioselective Synthesis of 4-Methyl-Substituted Dihydroisoquinolones-Reference-Cited by-同舟云学术

Rhodium(III)-Catalyzed C–H Activation: Ligand-Controlled Regioselective Synthesis of 4-Methyl-Substituted Dihydroisoquinolones

Published:2019-07-02 Issue:14 Volume:21 Page:5689-5693
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Barber Joyann S.¹,Scales Stephanie¹,Tran-Dubé Michelle¹,Wang Fen¹,Sach Neal W.¹,Bernier Louise¹,Collins Michael R.¹,Zhu JinJiang¹,McAlpine Indrawan J.¹,Patman Ryan L.¹^ORCID

Affiliation:

1. Pfizer Oncology Medicinal Chemistry, 10770 Science Center Drive, San Diego, California 92121, United States

Funder

Pfizer

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.9b02029

Reference43 articles.

1. Chemistry and Biology of the Tetrahydroisoquinoline Antitumor Antibiotics

2. Privileged scaffolds for library design and drug discovery

3. Design and synthesis of dihydroisoquinolones for fragment-based drug discovery (FBDD)

4. Opportunity Knocks: Organic Chemistry for Fragment-Based Drug Discovery (FBDD)

5. Tetrahydroisoquinolines in therapeutics: a patent review (2010-2015)

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