On-Resin Synthesis of Linear Aryl Thioether Containing Peptides and in-Solution Cyclization via Cysteine S<sub><i>N</i></sub>Ar Reaction-Reference-Cited by-同舟云学术

On-Resin Synthesis of Linear Aryl Thioether Containing Peptides and in-Solution Cyclization via Cysteine S_NAr Reaction

Published:2022-02-23 Issue:8 Volume:24 Page:1673-1677
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Li Jian¹^ORCID,Lai Weihong²,Pang Ao¹,Liu Lu¹,Ye Lianbao²,Xiong Xiao-Feng¹^ORCID

Affiliation:

1. Guangdong Key Laboratory of Chiral Molecule and Drug Discovery, School of Pharmaceutical Sciences, Sun Yat-sen University, 510006 Guangzhou, Guangdong, P. R. China

2. School of Pharmacy, Guangdong Pharmaceutical University, 510006 Guangzhou, Guangdong, P. R. China

Funder

National Natural Science Foundation of China

Natural Science Foundation of Guangdong Province

Guangdong Provincial Key Laboratory of Chiral Molecule and Drug Discovery

Key Reasearch and Development Program of Guangdong Province

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.2c00234

Reference41 articles.

1. Peptidomimetic toolbox for drug discovery

2. Orally Active Peptides: Is There a Magic Bullet?

3. Advances in oral peptide therapeutics

4. Proteolytically Stable Cyclic Decapeptide for Breast Cancer Cell Targeting

5. De novo Design of Selective Membrane‐Active Peptides by Enzymatic Control of Their Conformational Bias on the Cell Surface

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