Amide Formation: Choosing the Safer Carbodiimide in Combination with OxymaPure to Avoid HCN Release-Reference-Cited by-同舟云学术

Amide Formation: Choosing the Safer Carbodiimide in Combination with OxymaPure to Avoid HCN Release

Published:2021-08-23 Issue:17 Volume:23 Page:6900-6904
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Manne Srinivasa Rao¹,Luna Omar²³,Acosta Gerardo A.²³,Royo Miriam²³^ORCID,El-Faham Ayman⁴^ORCID,Orosz Gyorgy⁵,de la Torre Beatriz G.⁶^ORCID,Albericio Fernando¹²³^ORCID

Affiliation:

1. Peptide Science Laboratory, School of Chemistry and Physics, University of KwaZulu-Natal, Durban 4001, South Africa

2. Institute for Advanced Chemistry of Catalonia (IQAC−CSIC), 08034 Barcelona, Spain

3. CIBER-BBN, Networking Centre on Bioengineering, Biomaterials and Nanomedicine, and Department of Organic Chemistry, University of Barcelona, 08028 Barcelona, Spain

4. Department of Chemistry, Faculty of Science, Alexandria University, Ibrahimia, Alexandria 21321, Egypt

5. Luxembourg Bio Technologies, Ness Ziona 7403631, Israel

6. KwaZulu-Natal Research Innovation and Sequencing Platform (KRISP), School of Laboratory Medicine and Medical Sciences, College of Health Sciences, University of KwaZulu-Natal, Durban 4041, South Africa

Funder

H2020 Marie SkÅ?odowska-Curie Actions

National Research Foundation

PAVE

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.1c02466

Reference22 articles.

1. The Medicinal Chemist’s Toolbox: An Analysis of Reactions Used in the Pursuit of Drug Candidates