Mapping General Anesthetic Binding Site(s) in Human α1β3 γ-Aminobutyric Acid Type A Receptors with [3H]TDBzl-Etomidate, a Photoreactive Etomidate Analogue-Reference-Cited by-同舟云学术

Mapping General Anesthetic Binding Site(s) in Human α1β3 γ-Aminobutyric Acid Type A Receptors with [3H]TDBzl-Etomidate, a Photoreactive Etomidate Analogue

Published:2012-01-23 Issue:4 Volume:51 Page:836-847
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Chiara David C.,Dostalova Zuzana¹,Jayakar Selwyn S.,Zhou Xiaojuan¹,Miller Keith W.¹,Cohen Jonathan B.

Affiliation:

1. Department of Anesthesia, Critical Care, and Pain Medicine, Massachusetts General Hospital, Boston, Massachusetts 02114, United States

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi201772m

Reference46 articles.

1. Emerging molecular mechanisms of general anesthetic action

2. General anaesthesia: from molecular targets to neuronal pathways of sleep and arousal

3. Clinical and Molecular Pharmacology of Etomidate

4. Stereoselective Effects of Etomidate Optical Isomers on Gamma-aminobutyric Acid Type A Receptors and Animals

5. Gating Allosterism at a Single Class of Etomidate Sites on α1β2γ2L GABAA Receptors Accounts for Both Direct Activation and Agonist Modulation

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