A New Class of Nonsteroidal Aromatase Inhibitors: Design and Synthesis of Chromone and Xanthone Derivatives and Inhibition of the P450 Enzymes Aromatase and 17α-Hydroxylase/C17,20-Lyase-Reference-Cited by-同舟云学术

A New Class of Nonsteroidal Aromatase Inhibitors: Design and Synthesis of Chromone and Xanthone Derivatives and Inhibition of the P450 Enzymes Aromatase and 17α-Hydroxylase/C17,20-Lyase

Published:2001-01-24 Issue:5 Volume:44 Page:672-680
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Recanatini Maurizio¹,Bisi Alessandra¹,Cavalli Andrea¹,Belluti Federica¹,Gobbi Silvia¹,Rampa Angela¹,Valenti Piero¹,Palzer Martina¹,Palusczak Anja¹,Hartmann Rolf W.¹

Affiliation:

1. Department of Pharmaceutical Sciences, University of Bologna, Via Belmeloro 6, I-40126 Bologna, Italy, and Pharmaceutical and Medicinal Chemistry, Universität des Saarlandes, P.O. Box 15 11 50, D-66041 Saarbrücken, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000955s

Reference43 articles.

1. The Effect of an Aromatase Inhibitor, 4-Hydroxy-4-Androstene- 3,17-Dione, On Estrogen-Dependent Processes in Reproduction and Breast Cancer11

2. Estrone sulfatase versus estrone sulfotransferase in human breast cancer: potential clinical applications

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