1. Department
of Organic Chemistry, Stockholm University, Stockholm 10691, Sweden
2. RIA iMed, Medicinal Chemistry, AstraZeneca R&D, Mölndal 43183, Sweden
3. CVMD iMed, Medicinal Chemistry, AstraZeneca R&D, Mölndal 43183, Sweden
4. Departamento
de Química Orgánica I, Universidad del País Vasco/UPV-EHU, Manuel de Lardizabal 3, Donostia−San
Sebastián 20018, Spain