Metalloprotein-Catalyzed Click Reaction for In Situ Generation of a Potent Inhibitor-Reference-Cited by-同舟云学术

Metalloprotein-Catalyzed Click Reaction for In Situ Generation of a Potent Inhibitor

Published:2020-04-13 Issue:10 Volume:10 Page:5383-5392
ISSN:2155-5435
Container-title:ACS Catalysis
language:en
Short-container-title:ACS Catal.

Author:

Miyake Yuka¹²,Itoh Yukihiro¹²^ORCID,Suzuma Yoshinori²,Kodama Hidehiko²,Kurohara Takashi¹,Yamashita Yasunobu¹,Narozny Remy¹,Hanatani Yutaro¹,Uchida Shusaku³,Suzuki Takayoshi¹²⁴^ORCID

Affiliation:

1. The Institute of Scientific and Industrial Research (ISIR), Osaka University, Mihogaoka, Ibaraki-shi, Osaka 567-0047, Japan

2. Graduate School of Medical Science, Kyoto Prefectural University of Medicine, 1-5 Shimogamo-hangi-cho, Sakyo-ku, Kyoto 606-0823, Japan

3. Graduate School of Medicine, Kyoto University, 53 Shogoin Kawahara-cho, Sakyo-ku, Kyoto 606-8507, Japan

4. CREST, Japan Science and Technology Agency (JST), 4-1-8 Honcho, Kawaguchi, Saitama 332-0012, Japan

Funder

Ministry of Education, Culture, Sports, Science and Technology

Core Research for Evolutional Science and Technology

Japan Agency for Medical Research and Development

Publisher

American Chemical Society (ACS)

Subject

Catalysis,General Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acscatal.0c00369

Reference37 articles.

1. In situclick chemistry: from small molecule discovery to synthetic antibodies

2. In situ click chemistry: probing the binding landscapes of biological molecules

3. Flavonoids as RTK inhibitors and potential anticancer agents

4. Epitope Targeting of Tertiary Protein Structure Enables Target-Guided Synthesis of a Potent In-Cell Inhibitor of Botulinum Neurotoxin

5. Click Chemistry: Diverse Chemical Function from a Few Good Reactions

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