Covalent Inhibition Mechanism of Antidiabetic Drugs—Vildagliptin vs Saxagliptin
Author:
Affiliation:
1. School of Pharmaceutical Sciences, Sun Yat-sen University, Guangzhou 510006, P. R. China
2. Institute of Traditional Chinese Medicine & Natural Products, College of Pharmacy, Jinan University, Guangzhou 510632, P. R. China
Funder
Ministry of Science and Technology of the People's Republic of China
National Natural Science Foundation of China
Natural Science Foundation of Guangdong Province
Publisher
American Chemical Society (ACS)
Subject
Catalysis,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acscatal.8b05051
Reference67 articles.
1. Pharmacology and therapeutic implications of current drugs for type 2 diabetes mellitus
2. Dipeptidyl Peptidase IV and Its Inhibitors: Therapeutics for Type 2 Diabetes and What Else?
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4. Incretin therapies: highlighting common features and differences in the modes of action of glucagon‐like peptide‐1 receptor agonists and dipeptidyl peptidase‐4 inhibitors
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