From Serendipity to Rational Antituberculosis Drug Discovery of Mefloquine-Isoxazole Carboxylic Acid Esters-Reference-Cited by-同舟云学术

From Serendipity to Rational Antituberculosis Drug Discovery of Mefloquine-Isoxazole Carboxylic Acid Esters

Published:2009-10-28 Issue:22 Volume:52 Page:6966-6978
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mao Jialin¹,Yuan Hai²,Wang Yuehong¹,Wan Baojie¹,Pieroni Marco²,Huang Qingqing²,van Breemen Richard B.³,Kozikowski Alan P.²,Franzblau Scott G.¹

Affiliation:

1. Institute for Tuberculosis Research, College of Pharmacy

2. Drug Discovery Program, Department of Medicinal Chemistry and Pharmacognosy

3. Department of Medicinal Chemistry and Pharmacognosy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900340a

Reference11 articles.

1. WHO, WHO Report 2008 Global tuberculosis control - surveillance, planning, financing. 2008.

2. Fighting tuberculosis: An old disease with new challenges

3. HTS, Chemical Hybridization, and Drug Design Identify a Chemically Unique Antituberculosis Agent–Coupling Serendipity and Rational Approaches to Drug Discovery

4. Mao, J.; Yuan, H.; Wang, Y.; Wan, B.; Pak, D.; He, R.; Kozikowski, A. P; Franzblau, S. G.Synthesis and Antituberculosis Activity of Novel Mefloquine-Isoxazole Carboxylic Esters as Prodrugs (in preparation).

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