Modifications to the N-Terminus but Not the C-Terminus of Calcitonin Gene-Related Peptide(8-37) Produce Antagonists with Increased Affinity-Reference-Cited by-同舟云学术

Modifications to the N-Terminus but Not the C-Terminus of Calcitonin Gene-Related Peptide(8-37) Produce Antagonists with Increased Affinity

Published:2003-05-08 Issue:12 Volume:46 Page:2427-2435
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Smith D. David¹,Saha Shankar¹,Fang Guoyong¹,Schaffert Courtney¹,Waugh David J. J.¹,Zeng Wanyun¹,Toth Geza¹,Hulce Martin¹,Abel Peter W.¹

Affiliation:

1. Departments of Biomedical Sciences, Chemistry, and Pharmacology, Creighton University, 2500 California Plaza, Omaha, Nebraska 68178, and Isotope Laboratory, “B” Level, Biological Research Centre, Hungarian Academy of Sciences, P.O. Box 521, H-6701 Szeged, Hungary

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm020507f

Reference50 articles.

1. Neuroanatomical Localization, Pharmacological Characterization and Functions of CGRP, Related Peptides and Their Receptors

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