Further Definition of the D1 Dopamine Receptor Pharmacophore: Synthesis of trans-6,6a,7,8,9,13b-Hexahydro-5H-benzo[d]naphth[2,1-b]azepines as Rigid Analogues of β-Phenyldopamine-Reference-Cited by-同舟云学术

Further Definition of the D1 Dopamine Receptor Pharmacophore: Synthesis of trans-6,6a,7,8,9,13b-Hexahydro-5H-benzo[d]naphth[2,1-b]azepines as Rigid Analogues of β-Phenyldopamine

Published:1997-07-01 Issue:14 Volume:40 Page:2140-2147
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Negash Kitaw¹,Nichols David E.¹,Watts Val J.¹,Mailman Richard B.¹

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, School of Pharmacy and Pharmacal Sciences, Purdue University, West Lafayette, Indiana 47907, and UNC Neuroscience Center & Departments of Pharmacology and Psychiatry, University of North Carolina School of Medicine, Chapel Hill, North Carolina 27599-7250

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970157a

Reference26 articles.

1. Multiple receptors for dopamine

2. Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1

3. Identification of the 64K autoantigen in insulin-dependent diabetes as the GABA-synthesizing enzyme glutamic acid decarboxylase

4. Cloning of the gene for a human dopamine D5 receptor with higher affinity for dopamine than D1

5. Selective and stereospecific interactions of R-SK&F 38393 with [3H]piflutixol but not [3H]spiperone binding to striatal D1 and D2 dopamine receptors: Comparisons with SCH 23390

Cited by 13 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Asymmetric aminoarylation for the synthesis of trans-3-amino-4-aryltetrahydroquinolines: An access to aza-analogue of dihydrexidine;Tetrahedron;2022-01

2. Synthesis and dopaminergic activity of a series of new 1-aryl tetrahydroisoquinolines and 2-substituted 1-aryl-3-tetrahydrobenzazepines;Bioorganic Chemistry;2018-10

3. Tetrahydroisoquinolines functionalized with carbamates as selective ligands of D2 dopamine receptor;Journal of Molecular Modeling;2017-09

4. ChemInform Abstract: Further Definition of the D1 Dopamine Receptor Pharmacophore: Synthesis of trans-6,6a,7,8,9,13b-Hexahydro-5H-benzo(d)naphth(2,1-b) azepines as Rigid Analogues of β-Phenyldopamine.;ChemInform;2010-08-03

5. Diastereoselective Synthesis of 1,2-Disubstituted 2,3,4,5-Tetrahydro-1H-3-benzazepines by Means of the Stevens Rearrangement;European Journal of Organic Chemistry;2010-07-01