Recent Advances in the Design, Synthesis, and Biological Evaluation of Selective DYRK1A Inhibitors: A New Avenue for a Disease Modifying Treatment of Alzheimer’s?-Reference-Cited by-同舟云学术

Recent Advances in the Design, Synthesis, and Biological Evaluation of Selective DYRK1A Inhibitors: A New Avenue for a Disease Modifying Treatment of Alzheimer’s?

Published:2012-09-07 Issue:11 Volume:3 Page:857-872
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Smith Breland¹²,Medda Federico²,Gokhale Vijay³,Dunckley Travis⁴,Hulme Christopher¹²³

Affiliation:

1. Department of Chemistry & Biochemistry, the University of Arizona, Tucson, Arizona 85721, United States

2. BIO5 Oro Valley, the University of Arizona, 1580 East Hanley Boulevard, Oro Valley, Arizona 85737, United States

3. Department of Pharmacology & Toxicology, College of Pharmacy, University of Arizona, Tucson, Arizona 85721, United States

4. Neurogenomics Division, Translational Genomics Research Institute, Phoenix, Arizona 85013, United States

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/cn300094k

Reference124 articles.

1. Activation, regulation, and inhibition of DYRK1A

2. DYRK family of protein kinases: evolutionary relationships, biochemical properties, and functional roles

3. MNB/DYRK1A as a multiple regulator of neuronal development

4. Function and regulation of Dyrk1A: towards understanding Down syndrome

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