Design, Synthesis, and Evaluation of Conformationally Constrained Tongs, New Inhibitors of HIV-1 Protease Dimerization-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Conformationally Constrained Tongs, New Inhibitors of HIV-1 Protease Dimerization

Published:1999-02-27 Issue:6 Volume:42 Page:957-962
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bouras Ahmed¹,Boggetto Nicole¹,Benatalah Zohra¹,de Rosny Eve¹,Sicsic Sames¹,Reboud-Ravaux Michèle¹

Affiliation:

1. BIOCIS, URA-CNRS 1843, Faculté de Pharmacie, Université de Paris-sud, 5 rue J. B. Clément, F-92296 Châtenay-Malabry Cedex, France, and Laboratoire d'Enzymologie Moléculaire et Fonctionnelle, Département de Biologie Supramoléculaire et Cellulaire, Institut Jacques Monod, Universités de Paris VI et VII, 2 place Jussieu, F-75251 Paris Cedex 05, France

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9803976

Reference17 articles.

1. Role of human immunodeficiency virus type 1-specific protease in core protein maturation and viral infectivity

2. Thrombotic thrombocytopenic purpura and haemolytic uraemic syndrome in HIV-infected patients

3. Three-dimensional structure of aspartyl protease from human immunodeficiency virus HIV-1

4. Conserved Folding in Retroviral Proteases: Crystal Structure of Synthetic HIV-1 Protease

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