Optimized Inhibitors of Soluble Epoxide Hydrolase Improve in Vitro Target Residence Time and in Vivo Efficacy

Author:

Lee Kin Sing Stephen1,Liu Jun-Yan1,Wagner Karen M.1,Pakhomova Svetlana2,Dong Hua1,Morisseau Christophe1,Fu Samuel H.1,Yang Jun1,Wang Peng13,Ulu Arzu1,Mate Christina A.1,Nguyen Long V.1,Hwang Sung Hee1,Edin Matthew L.4,Mara Alexandria A.4,Wulff Heike5,Newcomer Marcia E.2,Zeldin Darryl C.4,Hammock Bruce D.1

Affiliation:

1. Department of Entomology and Nematology, UCD Comprehensive Cancer Center, University of California Davis, One Shields Avenue, Davis, California 95616, United States

2. Department of Biological Sciences, Louisiana State University, Baton Rouge, Louisiana 70803, United States

3. Department of Applied Chemistry, China Agricultural University, Beijing 100193, People’s Republic of China

4. Division of Intramural Research, National Institute of Environmental Health Sciences, National Institutes of Health, Research Triangle Park, North Carolina 27709, United States

5. Department of Pharmacology, University of California Davis, Davis, California 95616, United States

Funder

National Institute of Environmental Health Sciences

National Institute of Neurological Disorders and Stroke

Division of Biological Infrastructure

National Center for Research Resources

National Heart, Lung, and Blood Institute

U.S. Department of Energy

National Institute of Arthritis and Musculoskeletal and Skin Diseases

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Reference64 articles.

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2. Tolerating Diabetes: An Alternative Therapeutic Approach for Diabetic Neuropathy

3. Diabetic neuropathy—a review

4. Painful Diabetic Neuropathy: Epidemiology, Natural History, Early Diagnosis, and Treatment Options

5. Effects of treatments for symptoms of painful diabetic neuropathy: systematic review

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