SAR, Pharmacokinetics, Safety, and Efficacy of Glucokinase Activating 2-(4-Sulfonylphenyl)-N-thiazol-2-ylacetamides: Discovery of PSN-GK1-Reference-Cited by-同舟云学术

SAR, Pharmacokinetics, Safety, and Efficacy of Glucokinase Activating 2-(4-Sulfonylphenyl)-N-thiazol-2-ylacetamides: Discovery of PSN-GK1

Published:2008-06-28 Issue:14 Volume:51 Page:4340-4345
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bertram Lisa S.¹,Black Daniel¹,Briner Paul H.¹,Chatfield Rosemary¹,Cooke Andrew¹,Fyfe Matthew C. T.¹,Murray P. John¹,Naud Frédéric¹,Nawano Masao¹,Procter Martin J.¹,Rakipovski Günaj¹,Rasamison Chrystelle M.¹,Reynet Christine¹,Schofield Karen L.¹,Shah Vilas K.¹,Spindler Felix¹,Taylor Amanda¹,Turton Roy¹,Williams Geoffrey M.¹,Wong-Kai-In Philippe¹,Yasuda Kosuke¹

Affiliation:

1. (OSI) Prosidion, Windrush Court, Watlington Road, Oxford OX4 6LT, United Kingdom, (OSI) Pharmaceuticals, Inc., 2860 Wilderness Place, Boulder, Colorado 80301, Solvias AG, Klybeckstrasse 191, Postfach CH-4002 Basel, Switzerland, Mitsubishi Tanabe Pharma Corporation, 2-2-50 Kawagishi, Toda-shi, Saitama 335-8505, Japan, and Rheoscience A/S, Glerupvej 2, 2610 Rødovre, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm8003202

Reference38 articles.

1. New drug targets for type 2 diabetes and the metabolic syndrome

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3. A Comparison of Agents Used to Manage Type 2 Diabetes Mellitus

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