1-(2-Hydroxy-2-methyl-3-phenoxypropanoyl)indoline-4-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators-Reference-Cited by-同舟云学术

1-(2-Hydroxy-2-methyl-3-phenoxypropanoyl)indoline-4-carbonitrile Derivatives as Potent and Tissue Selective Androgen Receptor Modulators

Published:2014-03-10 Issue:6 Volume:57 Page:2462-2471
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Chekler Eugene L. Piatnitski¹,Unwalla Rayomond¹,Khan Taukeer A.¹,Tangirala Raghuram S.¹,Johnson Mark¹,St. Andre Michael¹,Anderson James T.¹,Kenney Thomas¹,Chiparri Sue¹,McNally Chris¹,Kilbourne Edward¹,Thompson Catherine¹,Nagpal Sunil¹,Weber Gregory¹,Schelling Scott¹,Owens Jane¹,Morris Carl A.¹,Powell Dennis¹,Verhoest Patrick R.¹,Gilbert Adam M.¹

Affiliation:

1. BioTherapeutics Medicinal Chemistry, Pfizer Global Research and Development, 200 Cambridgepark Drive, Cambridge, Massachusetts 02140, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401625b

Reference22 articles.

1. International Union of Pharmacology. LXV. The Pharmacology and Classification of the Nuclear Receptor Superfamily: Glucocorticoid, Mineralocorticoid, Progesterone, and Androgen Receptors

2. Chemistry and Structural Biology of Androgen Receptor

3. Selective androgen receptor modulators as function promoting therapies

4. Probing androgen receptor co-factor selectivity profiles: a chemical tool to determine cross-talk between androgen receptor and β-catenin in vivo

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