α,β-Unsaturated N-Acylpyrrole Peptidyl Derivatives: New Proteasome Inhibitors
Author:
Affiliation:
1. Department of Pharmaceutical Sciences and Biotechnology Center
2. Department of Chemistry and Center for Structural Diffractometry
3. Department of Biochemistry and Molecular Biology
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm100122e
Reference34 articles.
1. STRUCTURE AND FUNCTIONS OF THE 20S AND 26S PROTEASOMES
2. The Proteasome: Paradigm of a Self-Compartmentalizing Protease
3. The 26S Proteasome: A Molecular Machine Designed for Controlled Proteolysis
4. Crystal Structure of the 20 S Proteasome from the Archaeon T. acidophilum at 3.4 Å Resolution
5. MECHANISMS OF MHC CLASS I–RESTRICTED ANTIGEN PROCESSING
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