4‘-O-[2-(2-Fluoromalonyl)]-l-tyrosine: A Phosphotyrosyl Mimic for the Preparation of Signal Transduction Inhibitory Peptides-Reference-Cited by-同舟云学术

4‘-O-[2-(2-Fluoromalonyl)]-l-tyrosine: A Phosphotyrosyl Mimic for the Preparation of Signal Transduction Inhibitory Peptides

Published:1996-01-01 Issue:5 Volume:39 Page:1021-1027
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Burke, Terrence R.¹,Ye Bin¹,Akamatsu Miki¹,Ford, Harry¹,Yan Xinjian¹,Kole Hemanta K.¹,Wolf Gert¹,Shoelson Steven E.¹,Roller Peter P.¹

Affiliation:

1. Laboratory of Medicinal Chemistry, Building 37, Room 5C06, Division of Basic Sciences, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892, Laboratory of Clinical Physiology, Diabetes Unit, Gerontology Research Center, National Institute on Aging, National Institutes of Health, Baltimore, Maryland 21224, and Joslin Diabetes Center & Department of Medicine, Harvard Medical School, Boston, Massachusetts 02215

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm950621g

Reference33 articles.

1. A prelinary account of this work as been presented: Burke, T. R., Jr.; Ye, B.; Akamatsu, M.; Yan, X.; Kole, H. K.; Wolf, G.; Shoelson, S. E.; Roller, P. P. Non phosphorus-containing phosphotyrosyl mimetics amenable to prodrug derivatization and their use in solid-phase peptide synthesis of SH2 domain and phosphatase inhibitors. 209th National American Chemical Society Meeting, Anaheim, CA, April 2−7, 1995; MEDI 14.

2. Tyrosine protein kinase inhibition and cancer

3. Tyrosine Kinase Inhibition: An Approach to Drug Development

4. An Alternative to SH2 Domains for Binding Tyrosine-Phosphorylated Proteins

5. A phosphotyrosine interaction domain

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