A Novel Application of a Pd(0)-Catalyzed Nucleophilic Substitution Reaction to the Regio- and Stereoselective Synthesis of Lactam Analogues of the Epothilone Natural Products-Reference-Cited by-同舟云学术

A Novel Application of a Pd(0)-Catalyzed Nucleophilic Substitution Reaction to the Regio- and Stereoselective Synthesis of Lactam Analogues of the Epothilone Natural Products

Published:2000-08-26 Issue:37 Volume:122 Page:8890-8897
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Borzilleri Robert M.¹,Zheng Xiaoping¹,Schmidt Robert J.¹,Johnson James A.¹,Kim Soong-Hoon¹,DiMarco John D.¹,Fairchild Craig R.¹,Gougoutas Jack Z.¹,Lee Francis Y. F.¹,Long Byron H.¹,Vite Gregory D.¹

Affiliation:

1. Contribution from the Divisions of Discovery Chemistry, Oncology Drug Discovery, and Analytical Research and Development, The Bristol-Myers Squibb Pharmaceutical Research Institute, P.O. Box 4000, Princeton, New Jersey 08543-4000

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja001899n

Reference72 articles.

1. Epothilones: novel microtubule-stabilising agents

2. Activities of the Microtubule-stabilizing Agents Epothilones A and B with Purified Tubulin and in Cells Resistant to Paclitaxel (Taxol®)

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