Discovery of Covalent Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase, A Target for the Treatment of Malaria-Reference-Cited by-同舟云学术

Discovery of Covalent Inhibitors of Glyceraldehyde-3-phosphate Dehydrogenase, A Target for the Treatment of Malaria

Published:2014-09-02 Issue:17 Volume:57 Page:7465-7471
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Bruno Stefano¹²,Pinto Andrea³,Paredi Gianluca¹,Tamborini Lucia³,De Micheli Carlo³,La Pietra Valeria⁴,Marinelli Luciana⁴,Novellino Ettore⁴,Conti Paola³,Mozzarelli Andrea¹⁵

Affiliation:

1. Dipartimento di Farmacia and Centro Siteia.Parma, Università di Parma, Parco Area delle Scienze 23/A, 43124 Parma, Italy

2. Istituto di Bioscienze e Biorisorse, CNR, 80131 Napoli, Italy

3. Dipartimento di Scienze Farmaceutiche, Università degli Studi di Milano, Via Mangiagalli 25, 20133 Milano, Italy

4. Dipartimento di Farmacia, Università di Napoli Federico II, Via Montesano, 49, 80138 Napoli, Italy

5. Istituto Nazionale di Biostrutture e Biosistemi, 00136 Roma, Italy

Funder

Ministero degli Affari Esteri (MAE)

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm500747h

Reference35 articles.

1. GAPDH and Intermediary Metabolism

2. Snapshots of the Cystine Lyase C-DES during Catalysis

3. Protein crystal microspectrophotometry

4. Trapping of the Thioacylglyceraldehyde-3-phosphate Dehydrogenase Intermediate from Bacillus stearothermophilus

5. Anacardic acid derivatives as inhibitors of glyceraldehyde-3-phosphate dehydrogenase from Trypanosoma cruzi

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